Publication & Citation Trends
Publications
0 total
Discovery of PF-07265028, A Selective Small Molecule Inhibitor of Hematopoietic Progenitor Kinase 1 (HPK1) for the Treatment of Cancer.
Cited by 14
Semantic Scholar
Discovery of Clinical Candidate PF-06648671: A Potent γ-Secretase Modulator for the Treatment of Alzheimer's Disease.
Cited by 4
Semantic Scholar
SuFEx Activation with Ca(NTf2)2: A Unified Strategy to Access Sulfamides, Sulfamates, and Sulfonamides from S(VI) Fluorides OA
Cited by 70
Semantic Scholar
Optimization of Tubulysin Antibody–Drug Conjugates: A Case Study in Addressing ADC Metabolism OA
Cited by 62
Semantic Scholar
Design, Synthesis, and Cytotoxic Evaluation of Novel Tubulysin Analogues as ADC Payloads. OA
Cited by 30
Semantic Scholar
Discovery of Cytotoxic Dolastatin 10 Analogues with N-Terminal Modifications
Cited by 30
Semantic Scholar
Design of Pyridopyrazine-1,6-dione γ-Secretase Modulators that Align Potency, MDR Efflux Ratio, and Metabolic Stability. OA
Cited by 32
Semantic Scholar
Research Topics
Neuroscience and Neuropharmacology Research
(3)
Drug Transport and Resistance Mechanisms
(3)
Fluorine in Organic Chemistry
(3)
Sulfur-Based Synthesis Techniques
(3)
Synthesis and Catalytic Reactions
(3)
Affiliations
Pfizer (United States)