Publication & Citation Trends
Publications
0 total
The Discovery of GS-1291269: A Neutral Ketohexokinase (KHK) Inhibitor with an Unusual Thietane Amine Functional Group.
Cited by 1
Semantic Scholar
Discovery of Lanraplenib (GS-9876): A Once-Daily Spleen Tyrosine Kinase Inhibitor for Autoimmune Diseases. OA
Cited by 35
Semantic Scholar
Crystal structure of Syk in complex with GS-9876
Cited by 0
Semantic Scholar
Optimization of benzodiazepinones as selective inhibitors of the X-linked inhibitor of apoptosis protein (XIAP) second baculovirus IAP repeat (BIR2) domain.
Cited by 35
Semantic Scholar
Identification of 3-sulfonylindazole derivatives as potent and selective 5-HT(6) antagonists.
Cited by 19
Semantic Scholar
5-Piperazinyl-3-sulfonylindazoles as potent and selective 5-hydroxytryptamine-6 antagonists.
Cited by 53
Semantic Scholar
Synthesis, potency, and in vivo evaluation of 2-piperazin-1-ylquinoline analogues as dual serotonin reuptake inhibitors and serotonin 5-HT1A receptor antagonists.
Cited by 13
Semantic Scholar
1-Sulfonylindazoles as potent and selective 5-HT6 ligands.
Cited by 19
Semantic Scholar
Research Topics
Catalytic C–H Functionalization Methods
(6)
Sulfur-Based Synthesis Techniques
(4)
Asymmetric Synthesis and Catalysis
(3)
Cholinesterase and Neurodegenerative Diseases
(3)
Chemical synthesis and alkaloids
(3)
Affiliations
Pfizer (United States)
Princeton University
NOAA Chemical Sciences Laboratory